Fluconazole

Fluconazole – Broad-Spectrum Antifungal for Human and Veterinary Use

1. Introduction

Fluconazole is a triazole antifungal agent that works by inhibiting ergosterol synthesis, a key component of fungal cell membranes. It is widely used in human and veterinary medicine to treat fungal infections caused by Candida, Cryptococcus, Aspergillus, and others, offering strong efficacy and good oral bioavailability.

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2. Applications

2.1 In human pharmaceuticals

• Treats oral, esophageal, vaginal, gastrointestinal, skin, and systemic fungal infections

• Used as prophylaxis in immunocompromised patients, including HIV/AIDS cases

• Available in oral and intravenous forms

2.2 In veterinary medicine

• Effective against dermatophytosis, ear yeast infections, Malassezia, and Candida in pets

• Administered via oral or injectable forms for livestock and companion animals

• Long half-life allows for extended protection with fewer doses

3. Key advantages

• Excellent oral absorption, achieves high plasma concentration

• Broad antifungal spectrum

• High safety profile and minimal drug interactions

• Stable in tablets, powders, suspensions, and injectables

4. Product information

• Name: Fluconazole

• Form: White crystalline powder, odorless

• Purity: ≥ 99%

• Standards: USP / BP / EP

• Packaging: 1kg bags, 25kg fiber drums with PE liner

• Origin: China / India

• Storage: Store in a dry, cool place, protected from light, and keep container sealed

5. Conclusion

Fluconazole offers potent antifungal activity for both human and animal health. Its broad spectrum, high safety, and versatile formulation options make it a leading choice for antifungal drug development and clinical use.